Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50006711
TargetSerine protease 1(Bos taurus (bovine))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502661(CHEMBL4531752)
Affinity DataKi: <0.100nMAssay Description:Inhibition of bovine beta-trypsin using L-BAPNA as substrate preincubated for 5 mins followed by substrate addition and measured for 60 mins by color...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataKi:  3.20nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataKi:  6.10nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataKi:  7nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502659(CHEMBL4528256)
Affinity DataKi:  9.80nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataKi:  16nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataKi:  17nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502657(CHEMBL4589744)
Affinity DataKi:  23nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataKi:  24nMAssay Description:Inhibition of human neutrophil elastase using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502654(CHEMBL4470455)
Affinity DataKi:  51nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502660(CHEMBL4469546)
Affinity DataKi:  245nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataKi:  463nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human Cathepsin G using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Cathepsin G using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human alpha thrombin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human alpha thrombin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Cathepsin G using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human trypsin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human trypsin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human trypsin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human alpha thrombin using Boc-VPR-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human chymase expressed in Pichia pastoris using NleTDY-pNA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human chymase expressed in Pichia pastoris using NleTDY-pNA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human chymase expressed in Pichia pastoris using NleTDY-pNA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-C/Chymotrypsin-like protease CTRL-1/Chymotrypsinogen B/Chymotrypsinogen B2(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed