Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50009480
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 410nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50522742(CHEMBL4444522)
Affinity DataIC50: 7.00E+4nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50529225(CHEMBL4549736)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50529226(CHEMBL4444703)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50529225(CHEMBL4549736)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50529226(CHEMBL4444703)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50522742(CHEMBL4444522)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed