Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50009509
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529410(CHEMBL4463749)
Affinity DataEC50:  0.00510nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529411(CHEMBL4562635)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529412(CHEMBL4457592)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529413(CHEMBL4563672)
Affinity DataEC50:  0.00240nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529417(CHEMBL4548662)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataEC50:  0.00490nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529415(CHEMBL4588535)
Affinity DataEC50:  0.0140nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529416(CHEMBL4524446)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
United States Army Ccdc Chemical Biological Center

Curated by ChEMBL
LigandPNGBDBM50529414(CHEMBL4578287)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed