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Found 2 Enz. Inhib. hit(s) with all data for entry = 50010355
TargetAdenylate cyclase type 8(Homo sapiens (Human))
Kunming Medical University

Curated by ChEMBL
LigandPNGBDBM50537925(CHEMBL4644318)
Affinity DataEC50:  105nMAssay Description:Agonist activity at recombinant human AC8 expressed in human HEK293 cells assessed as fold increase in cAMP level by LANCE Ultra cAMP Detection kit m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 8(Homo sapiens (Human))
Kunming Medical University

Curated by ChEMBL
LigandPNGBDBM50010261((3R,4aR,5S,6S,6aS,10S,10aR,10bS)-3-ethenyl-6,10,10...)
Affinity DataEC50:  94nMAssay Description:Agonist activity at recombinant human AC8 expressed in human HEK293 cells assessed as fold increase in cAMP level by LANCE Ultra cAMP Detection kit m...More data for this Ligand-Target Pair