TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha/subunit alpha-11(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated platelet aggregationMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2/G(I)/G(S)/G(T) subunit beta-1(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair