Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50007961
TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514449(CHEMBL4171381)
Affinity DataIC50:  33nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50:  95nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(q) subunit alpha/subunit alpha-11(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50:  100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50:  100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM114291(8-(3,4,5-trihydroxy-6-keto-xanthen-9-yl)-1-naphtho...)
Affinity DataIC50:  130nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50246208(2-(3,4,5-trihydroxy-6-oxo-6H-xanthen-9-yl)cyclohex...)
Affinity DataIC50:  200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514448(CHEMBL4469620)
Affinity DataIC50:  200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514450(CHEMBL4443974)
Affinity DataIC50:  250nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50444748(Aminoquinuride)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM97335(7-amino-1,2,3,10-tetramethoxy-6,7-dihydro-5H-benzo...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514451(CHEMBL1967787)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed