Compile Data Set for Download or QSAR
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Found 36 Enz. Inhib. hit(s) with all data for entry = 50010476
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539339(CHEMBL4637769)
Affinity DataEC50:  252nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539350(CHEMBL4635551)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion preincubated with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539341(CHEMBL4632609)
Affinity DataEC50:  153nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539342(CHEMBL4641619)
Affinity DataEC50:  230nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539343(CHEMBL4639099)
Affinity DataEC50:  316nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539344(CHEMBL4647035)
Affinity DataEC50:  252nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539345(CHEMBL4645661)
Affinity DataEC50:  136nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539346(CHEMBL4641702)
Affinity DataEC50:  80nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539347(CHEMBL4639831)
Affinity DataEC50:  128nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539348(CHEMBL4647802)
Affinity DataEC50:  287nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539349(CHEMBL4636020)
Affinity DataEC50:  132nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539350(CHEMBL4635551)
Affinity DataEC50:  57nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539351(CHEMBL4635169)
Affinity DataEC50:  40nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539352(CHEMBL4636482)
Affinity DataEC50:  107nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539339(CHEMBL4637769)
Affinity DataEC50:  434nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539340(CHEMBL4640564)
Affinity DataEC50:  239nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539341(CHEMBL4632609)
Affinity DataEC50:  210nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539342(CHEMBL4641619)
Affinity DataEC50:  198nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539343(CHEMBL4639099)
Affinity DataEC50:  258nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539344(CHEMBL4647035)
Affinity DataEC50:  303nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539345(CHEMBL4645661)
Affinity DataEC50:  99nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539346(CHEMBL4641702)
Affinity DataEC50:  110nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539347(CHEMBL4639831)
Affinity DataEC50:  71nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539348(CHEMBL4647802)
Affinity DataEC50:  153nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539349(CHEMBL4636020)
Affinity DataEC50:  108nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539350(CHEMBL4635551)
Affinity DataEC50:  27nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539351(CHEMBL4635169)
Affinity DataEC50:  40nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539352(CHEMBL4636482)
Affinity DataEC50:  56nMAssay Description:Agonist activity at TLR7 in mouse BMDC cells assessed as immunostimulatory activity by measuring increase in IL6 secretion incubated for 18 hrs by EL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539339(CHEMBL4637769)
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 6 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539342(CHEMBL4641619)
Affinity DataEC50:  490nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 6 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539345(CHEMBL4645661)
Affinity DataEC50:  277nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 6 h...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539350(CHEMBL4635551)
Affinity DataEC50:  186nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 6 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539339(CHEMBL4637769)
Affinity DataEC50:  2.11E+3nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion preincubated with...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539342(CHEMBL4641619)
Affinity DataEC50:  909nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion preincubated with...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539345(CHEMBL4645661)
Affinity DataEC50:  585nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion preincubated with...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 7(Mus musculus)
Kagoshima University

Curated by ChEMBL
LigandPNGBDBM50539340(CHEMBL4640564)
Affinity DataEC50:  234nMAssay Description:Agonist activity at TLR7 in mouse RAW264.7 cells assessed as immunostimulatory activity by measuring increase in TNFalpha secretion incubated for 18 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed