Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50010488
LigandPNGBDBM50539512(CHEMBL4635689)
Affinity DataEC50:  0.700nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539509(CHEMBL4639259)
Affinity DataEC50:  1.5nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539502(CHEMBL4644943)
Affinity DataEC50:  2nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539506(CHEMBL4649443)
Affinity DataEC50:  2.60nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539508(CHEMBL4647214)
Affinity DataEC50:  2.70nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539507(CHEMBL4648903)
Affinity DataEC50:  2.90nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539504(CHEMBL4635759)
Affinity DataEC50:  3.90nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539505(CHEMBL4638287)
Affinity DataEC50:  4.60nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539511(CHEMBL4643151)
Affinity DataEC50:  8nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539510(CHEMBL4647502)
Affinity DataEC50:  8.20nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539503(CHEMBL4645958)
Affinity DataEC50:  11nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539501(CHEMBL4635181)
Affinity DataEC50:  30nMAssay Description:Transactivation of GAL4-fused human PPARdelta expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539513(CHEMBL4640515)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by semi-automatic patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539514(CHEMBL4649683)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by semi-automatic patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539510(CHEMBL4647502)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARgamma expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539509(CHEMBL4639259)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARgamma expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539507(CHEMBL4648903)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARgamma expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539510(CHEMBL4647502)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARalpha expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539509(CHEMBL4639259)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARalpha expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandPNGBDBM50539507(CHEMBL4648903)
Affinity DataEC50: >1.00E+5nMAssay Description:Transactivation of GAL4-fused human PPARalpha expressed in African green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed