Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50008533
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM247270(US9447029, 2-[2-(3-Pentyloxyphenyl)-ethylamino]-N,...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50520206(CHEMBL4291394)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM161090(US9051240, 2-[2-(3-Butoxyphenyl)-ethylamino]-N,N-d...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50520207(CHEMBL4555166)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50520205(CHEMBL4575754)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Southampton

Curated by ChEMBL
LigandPNGBDBM50520208(CHEMBL4463136)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed