Compile Data Set for Download or QSAR
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Found 120 Enz. Inhib. hit(s) with all data for entry = 50008545
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520310(CHEMBL4470864)
Affinity DataIC50:  2nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520310(CHEMBL4470864)
Affinity DataIC50:  2nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520316(CHEMBL4445758)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520316(CHEMBL4445758)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520305(CHEMBL4559976)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520309(CHEMBL4576800)
Affinity DataIC50:  4nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520309(CHEMBL4576800)
Affinity DataIC50:  4nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520305(CHEMBL4559976)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520303(CHEMBL4459830)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520303(CHEMBL4459830)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520310(CHEMBL4470864)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520310(CHEMBL4470864)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520304(CHEMBL4459627)
Affinity DataIC50:  7.90nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520304(CHEMBL4459627)
Affinity DataIC50:  8nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520304(CHEMBL4459627)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520304(CHEMBL4459627)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520301(CHEMBL4558167)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520321(CHEMBL4473192)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520301(CHEMBL4558167)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520321(CHEMBL4473192)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520312(CHEMBL4559463)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520312(CHEMBL4559463)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520309(CHEMBL4576800)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520309(CHEMBL4576800)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520306(CHEMBL4455385)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520306(CHEMBL4455385)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520326(CHEMBL4562412)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520324(CHEMBL4472149)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520326(CHEMBL4562412)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520324(CHEMBL4472149)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520317(CHEMBL4551058)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520307(CHEMBL4472196)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520317(CHEMBL4551058)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520307(CHEMBL4472196)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520320(CHEMBL4458380)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520320(CHEMBL4458380)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520318(CHEMBL4592883)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50322650((S)-2-(2-(2,2-diphenylethoxy)acetamido)-5-guanidin...)
Affinity DataIC50:  501nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520318(CHEMBL4592883)
Affinity DataIC50:  510nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50322650((S)-2-(2-(2,2-diphenylethoxy)acetamido)-5-guanidin...)
Affinity DataIC50:  540nMAssay Description:Antagonist at C3a receptor in human LAD2 cells assessed as inhibition of C3a-induced beta-hexosaminidase release preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520323(CHEMBL4439578)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520323(CHEMBL4439578)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520302(CHEMBL4470384)
Affinity DataIC50:  790nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520302(CHEMBL4470384)
Affinity DataIC50:  794nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50322650((S)-2-(2-(2,2-diphenylethoxy)acetamido)-5-guanidin...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50322650((S)-2-(2-(2,2-diphenylethoxy)acetamido)-5-guanidin...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520315(CHEMBL4444281)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520315(CHEMBL4444281)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520325(CHEMBL4530755)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50520308(CHEMBL4551118)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at C3a receptor in human MDM cells assessed as inhibition of C3a-induced intracellular calcium release preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
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