Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50010502
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539689(CHEMBL4642043)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539662(CHEMBL4641579)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]-ghrelin from human GHS-R1a stably expressed in HEK cell membrane measured after 60 mins by gamma counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539670(CHEMBL4632482)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539671(CHEMBL4641219)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539685(CHEMBL4649089)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539672(CHEMBL4640189)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539687(CHEMBL4635089)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539662(CHEMBL4641579)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539669(CHEMBL4649373)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539689(CHEMBL4642043)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539697(CHEMBL4636832)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539663(CHEMBL4632411)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539688(CHEMBL4638263)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539676(CHEMBL4639430)
Affinity DataEC50:  103nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539693(CHEMBL4646005)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50462127(CHEMBL4239086)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539662(CHEMBL4641579)
Affinity DataEC50:  123nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539695(CHEMBL4649741)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539681(CHEMBL4634029)
Affinity DataEC50:  166nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539690(CHEMBL4645314)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539677(CHEMBL4641428)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539696(CHEMBL4641503)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539675(CHEMBL4636565)
Affinity DataEC50:  299nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539673(CHEMBL4635725)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539691(CHEMBL4642179)
Affinity DataEC50:  410nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539689(CHEMBL4642043)
Affinity DataIC50: 460nMAssay Description:Displacement of [125I]-ghrelin from human GHS-R1a stably expressed in HEK cell membrane measured after 60 mins by gamma counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539686(CHEMBL4644587)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539674(CHEMBL4636849)
Affinity DataEC50:  560nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539694(CHEMBL4633635)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539685(CHEMBL4649089)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539697(CHEMBL4636832)
Affinity DataEC50:  660nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539679(CHEMBL4638731)
Affinity DataEC50:  719nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539666(CHEMBL4641372)
Affinity DataEC50:  740nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539692(CHEMBL4638676)
Affinity DataEC50:  740nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539678(CHEMBL4633947)
Affinity DataEC50:  769nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539680(CHEMBL4643496)
Affinity DataEC50:  895nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539687(CHEMBL4635089)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539663(CHEMBL4632411)
Affinity DataIC50: 960nMAssay Description:Displacement of [125I]-ghrelin from human GHS-R1a stably expressed in HEK cell membrane measured after 60 mins by gamma counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539685(CHEMBL4649089)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]-ghrelin from human GHS-R1a stably expressed in HEK cell membrane measured after 60 mins by gamma counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539695(CHEMBL4649741)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539665(CHEMBL4637486)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539693(CHEMBL4646005)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539690(CHEMBL4645314)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539698(CHEMBL4641449)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539688(CHEMBL4638263)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539687(CHEMBL4635089)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of [125I]-ghrelin from human GHS-R1a stably expressed in HEK cell membrane measured after 60 mins by gamma counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539663(CHEMBL4632411)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 2(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539696(CHEMBL4641503)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at human GPR109A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539668(CHEMBL4637505)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539664(CHEMBL4647314)
Affinity DataEC50: >3.70E+3nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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