TargetCannabinoid receptor 2(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in CHO cells incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human FAAH expressed in HEK293 cells using AMC arachidonyl amide as substrate pre-incubated for 50 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human FAAH expressed in HEK293 cells using AMC arachidonyl amide as substrate pre-incubated for 50 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human FAAH expressed in HEK293 cells using AMC arachidonyl amide as substrate pre-incubated for 50 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human FAAH expressed in HEK293 cells using AMC arachidonyl amide as substrate pre-incubated for 50 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human FAAH expressed in HEK293 cells using AMC arachidonyl amide as substrate pre-incubated for 50 mins followed by substrate addition ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of FAAH (unknown origin)More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate incubated for 45 mins by reverse-phase HPLC-b...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 9.60nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of rat FAAH expressed in HEK293 cells using AEA as substrate by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of FAAH in rat brain homogenate using 2-arachidonoyl-[3H]-glycerol as substrate by scintillation counting methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of rat FAAH expressed in HEK293 cells using AEA as substrate by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate incubated for 45 mins by reverse-phase HPLC-b...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of FAAH in OF1 albino mouse brain homogenate assessed as reduction in [3H]ethanolamine production using [3H]anandamide as substrateMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of FAAH in rat brain homogenate using [3H]AEA as substrateMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 492nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)
Curated by ChEMBL
Assam University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate incubated for 45 mins by reverse-phase HPLC-b...More data for this Ligand-Target Pair