Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50007118
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM31197(CHEMBL211045 | Nutlin-3 | med.21724, Compound 186)
Affinity DataIC50:  600nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506487(CHEMBL4441886)
Affinity DataIC50:  891nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506494(CHEMBL4585139)
Affinity DataIC50:  1.40E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506486(CHEMBL4518146)
Affinity DataIC50:  1.90E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506491(CHEMBL4521951)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506485(CHEMBL4460980)
Affinity DataIC50:  3.22E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506488(CHEMBL4474794)
Affinity DataIC50:  3.60E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506487(CHEMBL4441886)
Affinity DataIC50:  3.60E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506486(CHEMBL4518146)
Affinity DataIC50:  3.90E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506490(CHEMBL4460091)
Affinity DataIC50:  3.95E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506495(CHEMBL4448426)
Affinity DataIC50:  4.14E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506484(CHEMBL4530683)
Affinity DataIC50:  4.61E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506485(CHEMBL4460980)
Affinity DataIC50:  4.90E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506492(CHEMBL4436594)
Affinity DataIC50:  4.90E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506484(CHEMBL4530683)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506491(CHEMBL4521951)
Affinity DataIC50:  6.00E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506488(CHEMBL4474794)
Affinity DataIC50:  6.60E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506490(CHEMBL4460091)
Affinity DataIC50:  7.10E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506489(CHEMBL4592815)
Affinity DataIC50:  7.10E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM31197(CHEMBL211045 | Nutlin-3 | med.21724, Compound 186)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506496(CHEMBL4586161)
Affinity DataIC50:  1.03E+4nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506489(CHEMBL4592815)
Affinity DataIC50:  1.66E+4nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506491(CHEMBL4521951)
Affinity DataKd:  57nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506489(CHEMBL4592815)
Affinity DataKd:  99nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506484(CHEMBL4530683)
Affinity DataKd:  208nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506496(CHEMBL4586161)
Affinity DataKd:  109nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506494(CHEMBL4585139)
Affinity DataKd:  184nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506487(CHEMBL4441886)
Affinity DataKd:  26nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506485(CHEMBL4460980)
Affinity DataKd:  279nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506495(CHEMBL4448426)
Affinity DataKd:  181nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506489(CHEMBL4592815)
Affinity DataKd:  440nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506491(CHEMBL4521951)
Affinity DataKd:  370nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506490(CHEMBL4460091)
Affinity DataKd:  98nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506484(CHEMBL4530683)
Affinity DataKd:  641nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506490(CHEMBL4460091)
Affinity DataKd:  593nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506487(CHEMBL4441886)
Affinity DataKd:  221nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506485(CHEMBL4460980)
Affinity DataKd:  90nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506493(CHEMBL4453337)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50506492(CHEMBL4436594)
Affinity DataKd:  152nMAssay Description:Binding affinity to human MDM2 expressed in Escherichia coli expression system by using (FITC)-labeled p53 peptide based fluorescence polarization co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed