Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50013262
TargetMu-type opioid receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membrane incubated for 2.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Inhibition of sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membrane incubated for 2.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 165nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 238nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 253nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 269nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 402nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 506nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 573nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 573nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 694nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 835nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Huazhong University of Science and Technology
Curated by ChEMBL
Huazhong University of Science and Technology
Curated by ChEMBL
Affinity DataKi: 893nMAssay Description:Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation countin...More data for this Ligand-Target Pair

























