Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50011808
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551270(CHEMBL4776770)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551303(CHEMBL4755706)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551304(CHEMBL4796137)
Affinity DataIC50: 8nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551305(CHEMBL4750219)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551292(CHEMBL4758859)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551301(CHEMBL4791394)
Affinity DataIC50: 10nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551300(CHEMBL4756075)
Affinity DataIC50: 12nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551306(CHEMBL4796986)
Affinity DataIC50: 16nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551288(CHEMBL4796952)
Affinity DataIC50: 21nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551271(CHEMBL4747491)
Affinity DataIC50: 22nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551293(CHEMBL4749403)
Affinity DataIC50: 28nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551296(CHEMBL4795074)
Affinity DataIC50: 29nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551284(CHEMBL4754471)
Affinity DataIC50: 36nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551289(CHEMBL4749890)
Affinity DataIC50: 44nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551299(CHEMBL4749073)
Affinity DataIC50: 53nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551284(CHEMBL4754471)
Affinity DataIC50: 71nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551302(CHEMBL4791753)
Affinity DataIC50: 73nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551294(CHEMBL4795513)
Affinity DataIC50: 78nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551282(CHEMBL4751396)
Affinity DataIC50: 87nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551295(CHEMBL4796127)
Affinity DataIC50: 90nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551283(CHEMBL4777694)
Affinity DataIC50: 93nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551285(CHEMBL4755667)
Affinity DataIC50: 98nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataIC50: 106nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551280(CHEMBL4755685)
Affinity DataIC50: 108nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551298(CHEMBL4740899)
Affinity DataIC50: 108nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551271(CHEMBL4747491)
Affinity DataIC50: 109nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551289(CHEMBL4749890)
Affinity DataIC50: 126nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551276(CHEMBL4759383)
Affinity DataIC50: 138nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551278(CHEMBL4793358)
Affinity DataIC50: 150nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551275(CHEMBL4759851)
Affinity DataIC50: 154nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551274(CHEMBL4779839)
Affinity DataIC50: 162nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551277(CHEMBL4794106)
Affinity DataIC50: 169nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551279(CHEMBL4751651)
Affinity DataIC50: 172nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551272(CHEMBL4758654)
Affinity DataIC50: 172nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551297(CHEMBL4757805)
Affinity DataIC50: 208nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551285(CHEMBL4755667)
Affinity DataIC50: 266nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551277(CHEMBL4794106)
Affinity DataIC50: 269nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551291(CHEMBL4794713)
Affinity DataIC50: 284nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551281(CHEMBL4786547)
Affinity DataIC50: 296nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551290(CHEMBL4747773)
Affinity DataIC50: 313nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551273(CHEMBL4785799)
Affinity DataIC50: 341nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551280(CHEMBL4755685)
Affinity DataIC50: 351nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551290(CHEMBL4747773)
Affinity DataIC50: 352nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551275(CHEMBL4759851)
Affinity DataIC50: 414nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551273(CHEMBL4785799)
Affinity DataIC50: 423nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha-screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551283(CHEMBL4777694)
Affinity DataIC50: 426nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551272(CHEMBL4758654)
Affinity DataIC50: 434nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551282(CHEMBL4751396)
Affinity DataIC50: 505nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50551288(CHEMBL4796952)
Affinity DataIC50: 516nMAssay Description:Inhibition of full length human PLK1 using casein as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
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