Found 85 Enz. Inhib. hit(s) with all data for entry = 50010807 TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
3D Structure (crystal)Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 104nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 203nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 243nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 304nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 342nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 368nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 406nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 454nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 537nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 652nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 726nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
