Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50009336
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527521(CHEMBL4463788)
Affinity DataKd:  330nMAssay Description:Binding affinity to His-tagged PXR-LBD (unknown origin) expressed in Escherichia coli BL21 Gold by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527521(CHEMBL4463788)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527518(CHEMBL4566561)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527517(CHEMBL4467477)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527519(CHEMBL4465140)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527520(CHEMBL4455081)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50527522(CHEMBL4441887)
Affinity DataEC50:  1.70E+4nMAssay Description:Agonist activity at His-tagged PXR-LBD/SRC-1p (unknown origin) expressed in Escherichia coli BL21(DE3) by coactivator recruitment based Alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed