Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50011855
LigandPNGBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551826(CHEMBL4748416)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551833(CHEMBL4742674)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50424149(CHEMBL2312041)
Affinity DataIC50: 125nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551814(CHEMBL4793117)
Affinity DataIC50: 136nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551823(CHEMBL4744435)
Affinity DataIC50: 138nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551824(CHEMBL4777195)
Affinity DataIC50: 179nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551805(CHEMBL4756584)
Affinity DataIC50: 212nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551825(CHEMBL4751267)
Affinity DataIC50: 217nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551820(CHEMBL4753133)
Affinity DataIC50: 284nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551834(CHEMBL4747365)
Affinity DataIC50: 297nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50424148(CHEMBL2312042)
Affinity DataIC50: 302nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551802(CHEMBL4755512)
Affinity DataIC50: 317nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551822(CHEMBL4761891)
Affinity DataIC50: 336nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551827(CHEMBL4762536)
Affinity DataIC50: 347nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551804(CHEMBL4749849)
Affinity DataIC50: 365nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551807(CHEMBL4760687)
Affinity DataIC50: 387nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551829(CHEMBL4746914)
Affinity DataIC50: 389nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551806(CHEMBL4760707)
Affinity DataIC50: 424nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551803(CHEMBL4753763)
Affinity DataIC50: 463nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551835(CHEMBL4784720)
Affinity DataIC50: 481nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551813(CHEMBL4753274)
Affinity DataIC50: 543nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551832(CHEMBL4787388)
Affinity DataIC50: 568nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551821(CHEMBL4779721)
Affinity DataIC50: 569nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551830(CHEMBL4792182)
Affinity DataIC50: 594nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551828(CHEMBL4776648)
Affinity DataIC50: 684nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551831(CHEMBL4756407)
Affinity DataIC50: 765nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551817(CHEMBL4756090)
Affinity DataIC50: 787nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551808(CHEMBL4757691)
Affinity DataIC50: 854nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551812(CHEMBL4792573)
Affinity DataIC50: 874nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551816(CHEMBL4757020)
Affinity DataIC50: 952nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551819(CHEMBL4795871)
Affinity DataIC50: 1.07E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551815(CHEMBL4740420)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551811(CHEMBL4754416)
Affinity DataIC50: 1.25E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551818(CHEMBL4749358)
Affinity DataIC50: 1.45E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551810(CHEMBL4746256)
Affinity DataIC50: 7.53E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM50551809(CHEMBL4796780)
Affinity DataIC50: 9.42E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed