Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010946
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543625(CHEMBL3732444)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant full-length human aPKCzeta expressed in Sf21 insect cells using 5FAM-ERMRPRKRQGSVRRRV-NH2 as substrate in presence of ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C iota type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant full-length human aPKCiota using CREBtide as substrate incubated for 3 hrs in presence of ATP by kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543624(CHEMBL3732675)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using ERMRPRKRQGSVRRRV as substrate in presence of ATP by ADP Quest kit assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543617(CHEMBL4645321)
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543616(CHEMBL4647507)
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543614(CHEMBL4635556)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543618(CHEMBL4640268)
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543621(CHEMBL4633210)
Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543622(CHEMBL4649467)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta in presence of ATP at Km concentration by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543615(CHEMBL4648499)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543626(CHEMBL3729812)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant full-length human aPKCzeta expressed in Sf21 insect cells using 5FAM-ERMRPRKRQGSVRRRV-NH2 as substrate in presence of ATP a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C iota type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543619(CHEMBL4637651)
Affinity DataIC50: 4.08E+3nMAssay Description:Inhibition of recombinant full-length human aPKCiota in presence of ATP at Km concentration by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543620(CHEMBL4640910)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50543623(CHEMBL4638392)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of recombinant full-length human aPKCzeta using CREBtide as substrate incubated for 3 hrs in presence of ATP by Kinase Glo luminescent ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed