Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50010754
TargetMitogen-activated protein kinase 14(Mouse)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50541795(CHEMBL4634665)
Affinity DataKd:  2.51E+4nMAssay Description:Binding affinity to 6x-His tagged mouse recombinant p38alpha expressed in Escherichia coli Rosetta 2 (Novagen) cells by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 14(Mouse)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50541796(CHEMBL4634169)
Affinity DataKd:  5.78E+4nMAssay Description:Binding affinity to 6x-His tagged mouse recombinant p38alpha expressed in Escherichia coli Rosetta 2 (Novagen) cells by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 14(Mouse)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50541797(CHEMBL4646170)
Affinity DataKd:  1.12E+5nMAssay Description:Binding affinity to 6x-His tagged mouse recombinant p38alpha expressed in Escherichia coli Rosetta 2 (Novagen) cells by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)