Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50010755
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541803(CHEMBL4642490)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541802(CHEMBL4636138)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541800(CHEMBL4641092)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541799(CHEMBL4637022)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541798(CHEMBL4639113)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541800(CHEMBL4641092)
Affinity DataIC50: 50nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541801(CHEMBL4639560)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant His6Gb1-tagged HIF2alpha PAS B domain (240 to 350 residues)/human recombinant His6/FLAG-tagged ARNT PAS B domain (356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541803(CHEMBL4642490)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541802(CHEMBL4636138)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541801(CHEMBL4639560)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541799(CHEMBL4637022)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50541798(CHEMBL4639113)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIF2-alpha in human 786-0 cells cells harboring HRE-Luc2P reporter construct incubated for 48 hrs by ONE-Glo EX reagent based luminesce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed