Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50012241
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555835(CHEMBL4752175)
Affinity DataKi:  0.456nMAssay Description:Noncompetitive inhibition of human acetylcholinesterase assessed as affinity towards free enzyme using acetylthiocholine iodide as substrate measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555837(CHEMBL4747577)
Affinity DataKi:  8.30nMAssay Description:Mixed inhibition of human butyrylcholinesterase assessed as affinity towards free enzyme using butyrylthiocholine iodide as substrate measured by Ell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555837(CHEMBL4747577)
Affinity DataKi:  76nMAssay Description:Mixed inhibition of human butyrylcholinesterase assessed as affinity towards enzyme-substrate complex using butyrylthiocholine iodide as substrate me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555838(CHEMBL4752813)
Affinity DataIC50: 790nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555826(CHEMBL4745328)
Affinity DataIC50: 990nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555831(CHEMBL4747158)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555837(CHEMBL4747577)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555835(CHEMBL4752175)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555828(CHEMBL4759227)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555837(CHEMBL4747577)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555825(CHEMBL4745801)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555833(CHEMBL4795843)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555829(CHEMBL4753534)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555822(CHEMBL4789099)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555830(CHEMBL4749346)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555821(CHEMBL4758271)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555827(CHEMBL4790739)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555832(CHEMBL4748939)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555824(CHEMBL4743436)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555827(CHEMBL4790739)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555823(CHEMBL4761840)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555834(CHEMBL4762943)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555831(CHEMBL4747158)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555822(CHEMBL4789099)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555825(CHEMBL4745801)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555821(CHEMBL4758271)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555836(CHEMBL4762533)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555832(CHEMBL4748939)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555824(CHEMBL4743436)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555817(CHEMBL3621413)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555836(CHEMBL4762533)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555838(CHEMBL4752813)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555820(CHEMBL4745802)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555829(CHEMBL4753534)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555830(CHEMBL4749346)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555828(CHEMBL4759227)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555818(CHEMBL4758460)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555834(CHEMBL4762943)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555817(CHEMBL3621413)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555826(CHEMBL4745328)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555835(CHEMBL4752175)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555823(CHEMBL4761840)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555819(CHEMBL4756491)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555820(CHEMBL4745802)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of recombinant human Prolyl oligopeptidase expressed in Escherichia coli expression system using (Z)-Gly-Pro-p-nitroanilide as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555833(CHEMBL4795843)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555818(CHEMBL4758460)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50203126(Berberinechloride | 9,10-Dimethoxy-5,6-dihydro-[1,...)
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of recombinant human acetylcholinesterase using acetylthiocholine iodide as substrate preincubated with enzyme for 5 mins followed by subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555823(CHEMBL4761840)
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of recombinant human Prolyl oligopeptidase expressed in Escherichia coli expression system using (Z)-Gly-Pro-p-nitroanilide as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555826(CHEMBL4745328)
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of recombinant human Prolyl oligopeptidase expressed in Escherichia coli expression system using (Z)-Gly-Pro-p-nitroanilide as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Defense

Curated by ChEMBL
LigandPNGBDBM50555819(CHEMBL4756491)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human butyrylcholinesterase in plasma using butyrylthiocholineiodide as substrate preincubated with enzyme for 5 mins followed by subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
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