Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50012785
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560311(CHEMBL4756197)
Affinity DataIC50: 1nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560315(CHEMBL4763360)
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560326(CHEMBL4758563)
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560313(CHEMBL4762028)
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560319(CHEMBL4759758)
Affinity DataIC50: 7nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560323(CHEMBL4777937)
Affinity DataIC50: 7nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560317(CHEMBL4795123)
Affinity DataIC50: 8nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560324(CHEMBL4755015)
Affinity DataIC50: 9nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560318(CHEMBL4754348)
Affinity DataIC50: 21nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560312(CHEMBL4797614)
Affinity DataIC50: 22nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560325(CHEMBL4778549)
Affinity DataIC50: 26nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560316(CHEMBL4796205)
Affinity DataIC50: 34nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560321(CHEMBL4758961)
Affinity DataIC50: 73nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560314(CHEMBL4743141)
Affinity DataIC50: 79nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560322(CHEMBL4780682)
Affinity DataIC50: 90nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560320(CHEMBL4777252)
Affinity DataIC50: 107nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560310(CHEMBL4744881)
Affinity DataIC50: 5.00E+3nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50560310(CHEMBL4744881)
Affinity DataIC50: 5.00E+3nMAssay Description:Partial agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed