Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50012794
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50112347(CHEMBL3609327 | FRAX597)
Affinity DataIC50: 23nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560382(CHEMBL4777980)
Affinity DataIC50: 220nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560383(CHEMBL4779121)
Affinity DataIC50: 830nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560381(CHEMBL4747190)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560367(CHEMBL4748052)
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560368(CHEMBL4799887)
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560384(CHEMBL4743541)
Affinity DataIC50: 4.35E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560360(CHEMBL4779460)
Affinity DataIC50: 5.77E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560371(CHEMBL4761972)
Affinity DataIC50: 5.77E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560369(CHEMBL4764030)
Affinity DataIC50: 7.38E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560373(CHEMBL4755550)
Affinity DataIC50: 7.83E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560364(CHEMBL4761779)
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560375(CHEMBL4743990)
Affinity DataIC50: 9.56E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560366(CHEMBL4784170)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560370(CHEMBL4791897)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560365(CHEMBL4741943)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560374(CHEMBL4741285)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560363(CHEMBL4747878)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560380(CHEMBL4747628)
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560362(CHEMBL4791784)
Affinity DataIC50: 2.41E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560376(CHEMBL4793325)
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560372(CHEMBL4759481)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560377(CHEMBL4779690)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560378(CHEMBL4790502)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560379(CHEMBL4754223)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Harbin Medical University

Curated by ChEMBL
LigandPNGBDBM50560361(CHEMBL4752168)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed