Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50011344
TargetCystic fibrosis transmembrane conductance regulator(Human)
Rccs Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50546506(CHEMBL4764198)
Affinity DataEC50:  1.80E+3nMAssay Description:Potentiation of CFTR F508 deletion mutant (unknown origin) expressed in CFBE41o- cells coexpressing HS-YFP assessed as increase in intracellular cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
Rccs Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50546507(CHEMBL4746459)
Affinity DataEC50:  3.20E+3nMAssay Description:Potentiation of CFTR F508 deletion mutant (unknown origin) expressed in CFBE41o- cells coexpressing HS-YFP assessed as increase in intracellular cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed