Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50011392
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546677(CHEMBL4796102)
Affinity DataKi:  79nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546686(CHEMBL4795598)
Affinity DataKi:  794nMAssay Description:Antagonist activity at 5HT2C receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546686(CHEMBL4795598)
Affinity DataKi:  1.00E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546679(CHEMBL4780527)
Affinity DataKi:  1.00E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546682(CHEMBL4755344)
Affinity DataKi:  1.26E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546683(CHEMBL4741776)
Affinity DataKi:  1.59E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546678(CHEMBL4763861)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546682(CHEMBL4755344)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist activity at 5HT2C receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546680(CHEMBL4790230)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546685(CHEMBL4746138)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546684(CHEMBL4743625)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546681(CHEMBL4783824)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at 5HT2B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546683(CHEMBL4741776)
Affinity DataKi:  3.16E+3nMAssay Description:Antagonist activity at 5HT2C receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546678(CHEMBL4763861)
Affinity DataKi:  3.16E+3nMAssay Description:Antagonist activity at 5HT2C receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546677(CHEMBL4796102)
Affinity DataIC50:  6.31E+3nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) assessed as inhibition of 5HT-indued response by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM50546677(CHEMBL4796102)
Affinity DataEC50:  501nMAssay Description:Agonist activity at 5-HT2B receptor (unknown origin) by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Kalamazoo College

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataEC50:  0.0708nMAssay Description:Agonist activity at 5-HT2B receptor (unknown origin) by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed