Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50011399
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50546706(CHEMBL4797693)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546707(CHEMBL4778333)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546708(CHEMBL4791658)
Affinity DataEC50:  0.920nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546709(CHEMBL4753509)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546710(CHEMBL4796794)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546711(CHEMBL4751429)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546712(CHEMBL4748581)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546713(CHEMBL4752419)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546714(CHEMBL4799770)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546715(CHEMBL4791768)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546716(CHEMBL4742782)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546717(CHEMBL4781615)
Affinity DataEC50:  4nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546718(CHEMBL4743536)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546719(CHEMBL4746298)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546720(CHEMBL4740291)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546721(CHEMBL4756792)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546722(CHEMBL4749038)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546723(CHEMBL4785561)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546724(CHEMBL4787872)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546725(CHEMBL4744747)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546726(CHEMBL4796441)
Affinity DataEC50:  56nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546727(CHEMBL4743846)
Affinity DataEC50:  117nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetApelin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at human APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50546706(CHEMBL4797693)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed