Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50010926
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543457BDBM50543457(CHEMBL4635039)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543458BDBM50543458(CHEMBL4642307)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445383BDBM50445383(CHEMBL3104471)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543461BDBM50543461(CHEMBL4638346)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543459BDBM50543459(CHEMBL4643905)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543462BDBM50543462(CHEMBL4633010)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543463BDBM50543463(CHEMBL4638745)
Affinity DataIC50: 102nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543460BDBM50543460(CHEMBL4642313)
Affinity DataIC50: 135nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50543464BDBM50543464(CHEMBL4635150)
Affinity DataIC50: 155nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed