Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50012904
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50318701([(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50423649(CHEMBL2110363 | CHEMBL2413521 | SB-674042)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561403(CHEMBL4776564)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561427(CHEMBL4759509)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50412863(JNJ-10397049 | CHEMBL359632)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561443(CHEMBL4795679)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561446(CHEMBL4756004)
Affinity DataKi:  3.55E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50434481(CHEMBL2385133 | CHEMBL2385134 | CHEMBL2385132)
Affinity DataKi:  4.47E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561435(CHEMBL519512)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561449(CHEMBL4076997)
Affinity DataKi:  5.13E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561421(CHEMBL4788760)
Affinity DataKi:  5.37E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561434(CHEMBL4763441)
Affinity DataKi:  7.76E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561441(CHEMBL4799630)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561445(CHEMBL4759413)
Affinity DataKi:  8.91E+3nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561419(CHEMBL4752300)
Affinity DataKi:  1.17E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561454(CHEMBL4756045)
Affinity DataKi:  1.48E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561428(CHEMBL4761896)
Affinity DataKi:  1.48E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561436(CHEMBL4787509)
Affinity DataKi:  1.48E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561439(CHEMBL4790273)
Affinity DataKi:  1.51E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561417(CHEMBL4799045)
Affinity DataKi:  1.55E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561442(CHEMBL4758573)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561407(CHEMBL4761684)
Affinity DataKi:  1.78E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561426(CHEMBL4741048)
Affinity DataKi:  2.09E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561411(CHEMBL4753295)
Affinity DataKi:  2.14E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561462(CHEMBL4756829)
Affinity DataKi:  2.45E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561448(CHEMBL4793440)
Affinity DataKi:  2.45E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561432(CHEMBL4747508)
Affinity DataKi:  3.24E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561405(CHEMBL4753288)
Affinity DataKi:  3.31E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561460(CHEMBL4745747)
Affinity DataKi:  3.39E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561413(CHEMBL4750883)
Affinity DataKi:  4.37E+4nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561422(CHEMBL4757762)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561423(CHEMBL4764826)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561424(CHEMBL4759634)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561425(CHEMBL4752342)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561429(CHEMBL4797148)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561430(CHEMBL4758335)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561431(CHEMBL4746505)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561433(CHEMBL4776984)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561406(CHEMBL4740043)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561408(CHEMBL4789448)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561409(CHEMBL4746743)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561410(CHEMBL4784054)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561412(CHEMBL4747970)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561414(CHEMBL4757251)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561415(CHEMBL1418028)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561416(CHEMBL4794519)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561418(CHEMBL4776269)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561420(CHEMBL3456810)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561453(CHEMBL4756729)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Philipps-University

Curated by ChEMBL
LigandPNGBDBM50561455(CHEMBL4788750)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]-SB67404 from human orexin 1 receptor expressed in CHO cells incubated for 2 hrs by whole cell radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
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