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Found 18 Enz. Inhib. hit(s) with all data for entry = 50012329
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556595(CHEMBL4740154)
Affinity DataIC50:  0.320nMAssay Description:Antagonist activity at human H3 receptor expressed in HEK293 cells centrifuged for 3 mins followed by 60 mins incubation by LANCE Ultra cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556587(CHEMBL4791397)
Affinity DataIC50:  640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556588(CHEMBL4752838)
Affinity DataIC50:  640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556586(CHEMBL4781670)
Affinity DataIC50:  640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556585(CHEMBL4751314)
Affinity DataIC50:  640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556593(CHEMBL4751815)
Affinity DataIC50:  680nMAssay Description:Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells using p-Tyramine as substrate incubated for 15 mins by fluorescence meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556590(CHEMBL4778798)
Affinity DataIC50:  860nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556594(CHEMBL4750523)
Affinity DataIC50:  860nMAssay Description:Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells using p-Tyramine as substrate incubated for 15 mins by fluorescence meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556589(CHEMBL4758784)
Affinity DataIC50:  960nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556595(CHEMBL4740154)
Affinity DataIC50:  2.85E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation incubated for 24 hrs by ThT fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556584(CHEMBL4744947)
Affinity DataIC50:  5.06E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by ThT fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556583(CHEMBL4755924)
Affinity DataIC50:  7.05E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by ThT fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556581(CHEMBL4743941)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556582(CHEMBL4797501)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556580(CHEMBL4757329)
Affinity DataIC50:  4.88E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556591(CHEMBL4763495)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50086229(CHEMBL326815)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556592(CHEMBL4777813)
Affinity DataIC50:  2.46E+5nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed