TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 237nMAssay Description:Competitive binding affinity to human MDM2 assessed as displacement of p1-LC4f peptide by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKi: 461nMAssay Description:Competitive binding affinity to human MDM2 assessed as displacement of p3-BPf peptide by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 1.40E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 1.78E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 9.31E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 8.39E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 5.53E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 1.16E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 1.95E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 2.70E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 1.56E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 5.71E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 4.45E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 4.36E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 410nMAssay Description:Binding affinity to recombinant human MDM2 (25 to 111 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by fluores...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 9.29E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 3.10E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology
Curated by ChEMBL
Tokyo Institute Of Technology
Curated by ChEMBL
Affinity DataKd: 5.29E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair