Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50012111
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554287(CHEMBL4745237)
Affinity DataKi:  237nMAssay Description:Competitive binding affinity to human MDM2 assessed as displacement of p1-LC4f peptide by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554287(CHEMBL4745237)
Affinity DataKi:  461nMAssay Description:Competitive binding affinity to human MDM2 assessed as displacement of p3-BPf peptide by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554280(CHEMBL4740011)
Affinity DataKd:  1.40E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554281(CHEMBL4762612)
Affinity DataKd:  1.78E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554282(CHEMBL4746809)
Affinity DataKd:  9.31E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554283(CHEMBL4745447)
Affinity DataKd:  8.39E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554284(CHEMBL4788038)
Affinity DataKd:  5.53E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554285(CHEMBL4795921)
Affinity DataKd:  1.16E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554286(CHEMBL4798424)
Affinity DataKd:  1.95E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554278(CHEMBL4785007)
Affinity DataKd:  2.70E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554279(CHEMBL4742963)
Affinity DataKd:  1.56E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554281(CHEMBL4762612)
Affinity DataKd:  5.71E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554285(CHEMBL4795921)
Affinity DataKd:  4.45E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554286(CHEMBL4798424)
Affinity DataKd:  4.36E+5nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant in presence of 50 uM p53 peptide by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554287(CHEMBL4745237)
Affinity DataKd:  410nMAssay Description:Binding affinity to recombinant human MDM2 (25 to 111 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by fluores...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554279(CHEMBL4742963)
Affinity DataKd:  9.29E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554277(CHEMBL4791628)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Tokyo Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50554278(CHEMBL4785007)
Affinity DataKd:  5.29E+4nMAssay Description:Binding affinity to human MDM2 assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed