Found 6 Enz. Inhib. hit(s) with all data for entry = 50012144 TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
3D Structure (crystal)TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataEC50: 5.40E+3nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)
Curated by ChEMBL
National Research Council (Icb-Cnr)
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
