Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50011633
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM148264(US8962630, 74 | Ribociclib | LEE011 | Kisqali | 7-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549567(CHEMBL4793312)
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM148264(US8962630, 74 | Ribociclib | LEE011 | Kisqali | 7-...)
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549563(CHEMBL4789393)
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549560(CHEMBL4752087)
Affinity DataIC50: 28nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549565(CHEMBL4749923)
Affinity DataIC50: 28nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549568(CHEMBL4799064)
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549562(CHEMBL4796124)
Affinity DataIC50: 45nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549567(CHEMBL4793312)
Affinity DataIC50: 52nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549563(CHEMBL4789393)
Affinity DataIC50: 53nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549566(CHEMBL4743047)
Affinity DataIC50: 53nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549561(CHEMBL4800120)
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549568(CHEMBL4799064)
Affinity DataIC50: 64nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549560(CHEMBL4752087)
Affinity DataIC50: 64nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549578(CHEMBL4791807)
Affinity DataIC50: 93nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549564(CHEMBL4782842)
Affinity DataIC50: 121nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549577(CHEMBL4761061)
Affinity DataIC50: 143nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549575(CHEMBL4746355)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549566(CHEMBL4743047)
Affinity DataIC50: 169nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549565(CHEMBL4749923)
Affinity DataIC50: 268nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549576(CHEMBL4796853)
Affinity DataIC50: 315nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549562(CHEMBL4796124)
Affinity DataIC50: 369nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549580(CHEMBL4743521)
Affinity DataIC50: 379nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549564(CHEMBL4782842)
Affinity DataIC50: 391nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549579(CHEMBL4762979)
Affinity DataIC50: 523nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549561(CHEMBL4800120)
Affinity DataIC50: 666nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549573(CHEMBL4777302)
Affinity DataIC50: 861nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549574(CHEMBL4783734)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549571(CHEMBL4741644)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549572(CHEMBL4757913)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549570(CHEMBL4781000)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50549569(CHEMBL4784526)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed