Found 39 Enz. Inhib. hit(s) with all data for entry = 50013688 
Affinity DataIC50: 4.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human A2A expressed in human HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins followed by NECA s...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human A2A expressed in human HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins followed by NECA s...More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Antagonist activity at human A2A expressed in human HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins followed by NECA s...More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 131nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 149nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 312nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 733nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO-K1 cell membrane preincubated for 5 mins followed measured after 50 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-ZM241385 from human recombinant A2A receptor expressed in human HEK293 cell membrane preincubated for 5 mins and measured after ...More data for this Ligand-Target Pair
Affinity DataEC50: 524nMAssay Description:Antagonist activity at human A2A receptor on T-cells assessed as increase of IL-2 production preincubated for 1 hr followed by addition of T-cell act...More data for this Ligand-Target Pair
Affinity DataEC50: 376nMAssay Description:Antagonist activity at human A2A receptor on T-cells assessed as increase of IL-2 production preincubated for 1 hr followed by addition of T-cell act...More data for this Ligand-Target Pair
Affinity DataEC50: 165nMAssay Description:Antagonist activity at human A2A receptor on T-cells assessed as increase of IL-2 production preincubated for 1 hr followed by addition of T-cell act...More data for this Ligand-Target Pair
