Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50035728
TargetDihydrofolate reductase(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50367055(4-Aminofolic acid | 4-Aminopteroic acid | Aminopte...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50023405(3-(Carboxymethyl-{4-[(2,4-diamino-pteridin-6-ylmet...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50023404(5-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-methyl-ami...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50023406(5-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-amino]-ben...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Mouse)
Institute

Curated by ChEMBL
LigandPNGBDBM50023408(2-{3-[(2,4-Diamino-pteridin-6-ylmethyl)-amino]-ben...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against dihydrofolate reductase(DHFR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed