Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50012419
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557516(CHEMBL4787347)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557512(CHEMBL4779775)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557516(CHEMBL4787347)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557516(CHEMBL4787347)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557513(CHEMBL4795739)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557513(CHEMBL4795739)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557513(CHEMBL4795739)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557514(CHEMBL4779296)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557517(CHEMBL4760082)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557514(CHEMBL4779296)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557517(CHEMBL4760082)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557517(CHEMBL4760082)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557514(CHEMBL4779296)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557515(CHEMBL4744219)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557512(CHEMBL4779775)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557511(CHEMBL4764017)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557512(CHEMBL4779775)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557515(CHEMBL4744219)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptor by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557515(CHEMBL4744219)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557511(CHEMBL4764017)
Affinity DataKi:  369nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557511(CHEMBL4764017)
Affinity DataKi:  865nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as inhibition of forskolin-stimulated cAMP level at 500 nM stimulated for 30 mins followed by Eu-...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins followed by Eu-cAMP tracer ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557517(CHEMBL4760082)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins followed by Eu-cAMP tracer ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557516(CHEMBL4787347)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins followed by Eu-cAMP tracer ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557514(CHEMBL4779296)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins followed by Eu-cAMP tracer ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50557513(CHEMBL4795739)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at rat brain CB1 receptor assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins followed by Eu-cAMP tracer ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cells assessed as decrease in forskolin-stimulated cAMP level stimulated for 30 mins follo...More data for this Ligand-Target Pair