Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50014600
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577843(CHEMBL4853460)
Affinity DataKi:  36nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577843(CHEMBL4853460)
Affinity DataKi:  47nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50531967(Pugnac)
Affinity DataKi:  50nMAssay Description:Inhibition of OGA (unknown origin) using pNP-O-GlcNAc as substrate assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577842(CHEMBL4866781)
Affinity DataKi:  83nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577838(CHEMBL4874886)
Affinity DataKi:  125nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577836(CHEMBL4861823)
Affinity DataKi:  130nMAssay Description:Inhibition of HexA/HexB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577840(CHEMBL4864246)
Affinity DataKi:  154nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577837(CHEMBL4875285)
Affinity DataKi:  155nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577838(CHEMBL4874886)
Affinity DataKi:  167nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577842(CHEMBL4866781)
Affinity DataKi:  170nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577836(CHEMBL4861823)
Affinity DataKi:  190nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit alpha(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577836(CHEMBL4861823)
Affinity DataKi:  205nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577839(CHEMBL4851727)
Affinity DataKi:  270nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577837(CHEMBL4875285)
Affinity DataKi:  332nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577839(CHEMBL4851727)
Affinity DataKi:  413nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577840(CHEMBL4864246)
Affinity DataKi:  506nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577840(CHEMBL4864246)
Affinity DataKi:  509nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577844(CHEMBL402605)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of OGA (unknown origin) using pNP-O-GlcNAc as substrate assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577841(CHEMBL4845911)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-hexosaminidase(Bovine)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577841(CHEMBL4845911)
Affinity DataKi:  3.00E+4nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed