Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50014474
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576685(CHEMBL4871128)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of Escherichia coli DsbA using DOTA/Eu(III)-CQQGFDGTQNSCK-MCA as substrate in presence of oxidized glutathione measured by fluorescence an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576685(CHEMBL4871128)
Affinity DataKd:  2.74E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576683(CHEMBL4854940)
Affinity DataKd:  4.03E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576682(CHEMBL4855609)
Affinity DataKd:  4.60E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576684(CHEMBL4848780)
Affinity DataKd:  5.31E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576679(CHEMBL4851994)
Affinity DataKd:  8.20E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576676(CHEMBL4868312)
Affinity DataKd:  8.30E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576686(CHEMBL4875684)
Affinity DataKd:  9.78E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576681(CHEMBL4846499)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576677(CHEMBL4877192)
Affinity DataKd:  1.10E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576680(CHEMBL4860222)
Affinity DataKd:  1.14E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50576678(CHEMBL4852788)
Affinity DataKd:  2.30E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed