Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50014477
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524064(US11136336, Example 15)
Affinity DataIC50: 9nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524060(US11136336, Example 11)
Affinity DataIC50: 10nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524041(US11136336, Example 1 | 3-({3-[(2S)-2-(4-chlorophe...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524061(US11136336, Example 12)
Affinity DataIC50: 15nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524065(US11136336, Example 16)
Affinity DataIC50: 16nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524052(US11136336, Example 3)
Affinity DataIC50: 19nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524062(US11136336, Example 13)
Affinity DataIC50: 37nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524055(US11136336, Example 6)
Affinity DataIC50: 48nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524057(US11136336, Example 8)
Affinity DataIC50: 56nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM524058(US11136336, Example 9)
Affinity DataIC50: 78nMAssay Description:Antagonist activity against human TRPA1 expressed in HEK293K cells assessed as inhibition of AITC-induced intracellular calcium accumulation measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed