Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50013540
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567201BDBM50567201(CHEMBL4875501)
Affinity DataKi:  5.70E+4nMAssay Description:Competitive inhibition of SARS CoV-2 main protease using varying concentrations of DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by Dixon plot anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567201BDBM50567201(CHEMBL4875501)
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567181BDBM50567181(CHEMBL4868572)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567182BDBM50567182(CHEMBL4859153)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567183BDBM50567183(CHEMBL4846937)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567184BDBM50567184(CHEMBL4873791)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567185BDBM50567185(CHEMBL4871930)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567186BDBM50567186(CHEMBL4855260)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567187BDBM50567187(CHEMBL4864163)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567188BDBM50567188(CHEMBL4867088)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567189BDBM50567189(CHEMBL4872397)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567190BDBM50567190(CHEMBL4851348)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567191BDBM50567191(CHEMBL4851196)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567192BDBM50567192(CHEMBL4876522)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567193BDBM50567193(CHEMBL4858748)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567194BDBM50567194(CHEMBL4848940)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567195BDBM50567195(CHEMBL4847752)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567196BDBM50567196(CHEMBL4873945)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567197BDBM50567197(CHEMBL4846266)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567198BDBM50567198(CHEMBL4877763)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567199BDBM50567199(CHEMBL4877806)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50567200BDBM50567200(CHEMBL4873357)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SARS CoV-2 main protease using DABCYL-KTSAVLQ1SGFRKM-E(EDANS)-NH2 as substrate by FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed