Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50015459
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586775BDBM50586775(CHEMBL5087398)
Affinity DataIC50: 12nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586774BDBM50586774(CHEMBL5082392)
Affinity DataIC50: 63nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586771BDBM50586771(CHEMBL5091645)
Affinity DataIC50: 123nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586776BDBM50586776(CHEMBL5091627)
Affinity DataIC50: 129nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586773BDBM50586773(CHEMBL5082440)
Affinity DataIC50: 140nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586772BDBM50586772(CHEMBL5086489)
Affinity DataIC50: 166nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50586770BDBM50586770(CHEMBL4454763)
Affinity DataIC50: 850nMAssay Description:Inhibition of human NEK1 using myelin basic protein as substrate assessed as residual activity in presence of [gamma-33P]-ATP by radiometric hotspot ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed