Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50015271
Affinity DataKd: 27nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 33nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 43nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 49nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 68nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 85nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 102nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 132nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 152nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based direct binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 383nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 758nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 780nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 910nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 2.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 2.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.80E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Affinity DataKd: 3.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 3.70E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Affinity DataKd: 4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 4.10E+3nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) interaction assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution ass...More data for this Ligand-Target Pair
Affinity DataKd: 4.70E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.00E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.10E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.40E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.50E+3nMAssay Description:Binding affinity to Keap1 (unknown origin) at R415 assessed as dissociation constant by surface plasmon resonance based inhibition-in-solution assayMore data for this Ligand-Target Pair

















3D Structure (crystal)











