Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50017644
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603651(CHEMBL5172363)
Affinity DataKi:  580nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603644(CHEMBL5207990)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603645(CHEMBL5201753)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataKi:  1.31E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50461615(CHEMBL4228875)
Affinity DataKi:  2.45E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50461633(CHEMBL4227896)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603650(CHEMBL5185370)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603640(CHEMBL5171518)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603652(CHEMBL5183927)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50241218(CHEMBL4103395)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603639(CHEMBL5170166)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603642(CHEMBL5175138)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603647(CHEMBL5171248)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50241228(CHEMBL4093689)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603643(CHEMBL5209213)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603631(CHEMBL5182693)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603641(CHEMBL5198422)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603646(CHEMBL5172565)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603637(CHEMBL5204768)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603628(CHEMBL5206465)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603629(CHEMBL5200147)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603649(CHEMBL5204288)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603626(CHEMBL5179904)
Affinity DataKi:  9.90E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603630(CHEMBL5201688)
Affinity DataKi:  9.90E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603634(CHEMBL5185703)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603653(CHEMBL5181063)
Affinity DataKi:  1.01E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603627(CHEMBL5195308)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603625(CHEMBL5204977)
Affinity DataKi:  1.22E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603635(CHEMBL5194961)
Affinity DataKi:  1.34E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603624(CHEMBL5181135)
Affinity DataKi:  1.53E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603621(CHEMBL5207403)
Affinity DataKi:  1.57E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603636(CHEMBL5187627)
Affinity DataKi:  1.62E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603648(CHEMBL5176385)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603620(CHEMBL5199338)
Affinity DataKi:  1.93E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603638(CHEMBL5201833)
Affinity DataKi:  2.03E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603622(CHEMBL5185184)
Affinity DataKi:  2.23E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603619(CHEMBL5175620)
Affinity DataKi:  2.54E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603656(CHEMBL5201604)
Affinity DataKi:  2.66E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603633(CHEMBL5198521)
Affinity DataKi:  2.76E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603623(CHEMBL5189561)
Affinity DataKi:  2.87E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50241217(CHEMBL4099998)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603632(CHEMBL5199878)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603618(CHEMBL5195388)
Affinity DataKi:  4.14E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603654(CHEMBL5196499)
Affinity DataKi:  4.67E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603655(CHEMBL5185364)
Affinity DataKi:  8.88E+4nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50603657(CHEMBL5203518)
Affinity DataKi:  2.53E+5nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed