Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50017660
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603782BDBM50603782(CHEMBL4596414)
Affinity DataIC50: 0.0810nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602542BDBM50602542(CHEMBL4594870)
Affinity DataIC50: 0.0860nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602545BDBM50602545(CHEMBL4596647)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603794BDBM50603794(CHEMBL5184737)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603779BDBM50603779(CHEMBL3558756)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603788BDBM50603788(CHEMBL5171874)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603795BDBM50603795(CHEMBL5175270)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602544BDBM50602544(CHEMBL4594757)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603793BDBM50603793(CHEMBL5199542)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603792BDBM50603792(CHEMBL5176188)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603781BDBM50603781(CHEMBL4596941)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603789BDBM50603789(CHEMBL5183942)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603783BDBM50603783(CHEMBL4595806)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603790BDBM50603790(CHEMBL5191563)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603796BDBM50603796(CHEMBL5204190)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603787BDBM50603787(CHEMBL4597308)
Affinity DataIC50: 0.710nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603780BDBM50603780(CHEMBL4596992)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603791BDBM50603791(CHEMBL5179302)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603786BDBM50603786(CHEMBL4595664)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602543BDBM50602543(CHEMBL4598338)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033762BDBM50033762(Gallinamide A)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603784BDBM50603784(CHEMBL4595223)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603797BDBM50603797(CHEMBL5202965)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603785BDBM50603785(CHEMBL4595559)
Affinity DataIC50: 5nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of California San Diego

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50603798BDBM50603798(CHEMBL5199098)
Affinity DataIC50: 30nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate addition by fluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed