Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50016264
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50121400(CHEMBL3616752)
Affinity DataEC50:  0.0190nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593638(CHEMBL5194540)
Affinity DataEC50:  0.0650nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593639(CHEMBL5191858)
Affinity DataEC50:  0.132nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593643(CHEMBL5199198)
Affinity DataEC50:  0.135nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593644(CHEMBL5193167)
Affinity DataEC50:  0.158nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593640(CHEMBL5175517)
Affinity DataEC50:  0.170nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593641(CHEMBL5180864)
Affinity DataEC50:  0.204nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593642(CHEMBL5179465)
Affinity DataEC50:  0.209nMAssay Description:Activation of GLP-1 receptor (unknown origin) expressed in CHO-K1 cells assessed as increase in cAMP accumulation by time-resolved fluorescence reson...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50121400(CHEMBL3616752)
Affinity DataKd:  441nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593643(CHEMBL5199198)
Affinity DataKd:  532nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593641(CHEMBL5180864)
Affinity DataKd:  700nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593640(CHEMBL5175517)
Affinity DataKd:  911nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593639(CHEMBL5191858)
Affinity DataKd:  994nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593642(CHEMBL5179465)
Affinity DataKd:  1.46E+3nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593644(CHEMBL5193167)
Affinity DataKd:  1.49E+3nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50593638(CHEMBL5194540)
Affinity DataKd:  3.75E+3nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China State Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50240819(CHEMBL4084119)
Affinity DataKd:  6.27E+3nMAssay Description:Binding affinity to GLP-1 receptor (unknown origin) assessed as equlibrium constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed