Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50016266
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593659BDBM50593659(CHEMBL5207265)
Affinity DataEC50:  64nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593660BDBM50593660(CHEMBL5170235)
Affinity DataEC50:  90nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593653BDBM50593653(CHEMBL5185974)
Affinity DataEC50:  97nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593654BDBM50593654(CHEMBL5204436)
Affinity DataEC50:  142nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593650BDBM50593650(CHEMBL5169533)
Affinity DataEC50:  199nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593656BDBM50593656(CHEMBL5183971)
Affinity DataEC50:  208nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593657BDBM50593657(CHEMBL5187574)
Affinity DataEC50:  294nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593658BDBM50593658(CHEMBL5193733)
Affinity DataEC50:  341nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593652BDBM50593652(CHEMBL5188066)
Affinity DataEC50:  419nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593649BDBM50593649(CHEMBL5202253)
Affinity DataEC50:  444nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593651BDBM50593651(CHEMBL5186902)
Affinity DataEC50:  496nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593655BDBM50593655(CHEMBL5209256)
Affinity DataEC50:  637nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593661BDBM50593661(CHEMBL2346820)
Affinity DataEC50:  764nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Human)
Chemical Works of Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50593648BDBM50593648(CHEMBL5209395)
Affinity DataEC50:  771nMAssay Description:Positive allosteric modulation of GABA-B receptor (unknown origin) assessed as stimulation of [35S]GTPgammaS binding by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed