Compile Data Set for Download or QSAR
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Found 104 Enz. Inhib. hit(s) with all data for entry = 50017777
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50254013(3-(4-Amino-3-methylbenzyl)-7-(2-furyl)-3H-[1,2,3]t...)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604937(CHEMBL5171906)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604939(CHEMBL5201523)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604938(CHEMBL5189051)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604941(CHEMBL5186576)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604945(CHEMBL5188801)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604949(CHEMBL5195323)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604936(CHEMBL5194232)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604940(CHEMBL5196802)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604935(CHEMBL5173073)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604943(CHEMBL5200632)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604942(CHEMBL5179765)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604944(CHEMBL5188108)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604946(CHEMBL5179716)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604947(CHEMBL5189321)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604950(CHEMBL5204735)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604939(CHEMBL5201523)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]DPCPX from human A1AR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604930(CHEMBL5190722)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604926(CHEMBL5193403)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604932(CHEMBL5208818)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604928(CHEMBL5202005)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604929(CHEMBL5205560)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604948(CHEMBL5171672)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604925(CHEMBL5199428)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604912(CHEMBL5169338)
Affinity DataKi:  276nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604920(CHEMBL5200340)
Affinity DataKi:  295nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604911(CHEMBL5197839)
Affinity DataKi:  301nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604915(CHEMBL5169828)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604933(CHEMBL5190589)
Affinity DataKi:  378nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604919(CHEMBL5176483)
Affinity DataKi:  436nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604925(CHEMBL5199428)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]DPCPX from human A1AR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604939(CHEMBL5201523)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]DPCPX from human A2BAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604916(CHEMBL5202905)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604914(CHEMBL5205993)
Affinity DataKi:  618nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604945(CHEMBL5188801)
Affinity DataKi:  641nMAssay Description:Displacement of [3H]DPCPX from human A1AR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604910(CHEMBL5207324)
Affinity DataKi:  778nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604917(CHEMBL5209296)
Affinity DataKi:  863nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604921(CHEMBL5201509)
Affinity DataKi:  863nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604927(CHEMBL5203443)
Affinity DataKi:  974nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604909(CHEMBL5194109)
Affinity DataKi:  1.56E+3nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604923(CHEMBL5184684)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604913(CHEMBL5192939)
Affinity DataKi:  1.83E+3nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604945(CHEMBL5188801)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]DPCPX from human A2BAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604918(CHEMBL5170997)
Affinity DataKi:  2.54E+3nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604931(CHEMBL5185100)
Affinity DataKi:  3.59E+3nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604922(CHEMBL5190098)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604924(CHEMBL5171122)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH5826 from human A2AAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604939(CHEMBL5201523)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]HEMADO from human A3AR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604925(CHEMBL5199428)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]HEMADO from human A3AR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50604925(CHEMBL5199428)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A2BAR incubated for 60 mins by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
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