Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50017844
TargetDual specificity mitogen-activated protein kinase kinase 3(Human)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKd: 71nMAssay Description:Binding affinity to CM5 chip immobilized human MKK3 (20 to 347 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constants,...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 3(Human)
Fudan University
Curated by ChEMBL
Fudan University
Curated by ChEMBL
Affinity DataKon: 0.00361M-1s-1Assay Description:Binding affinity to CM5 chip immobilized human MKK3 (20 to 347 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant, ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
