Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50017227
TargetAmine oxidase [flavin-containing] A(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 16nMAssay Description:Inhibition of rat brain MAOB using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 41nMAssay Description:Inhibition of rat brain MAOB using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 41nMAssay Description:Inhibition of rat brain MAOB using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 51nMAssay Description:Inhibition of rat brain MAOA using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 51nMAssay Description:Inhibition of rat brain MAOA using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 95nMAssay Description:Inhibition of human recombinant MAOB using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600361(CHEMBL5171345)
Affinity DataIC50: 140nMAssay Description:Inhibition of rat brain MAOA using kynuramine substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600362(CHEMBL5187434)
Affinity DataKi:  435nMAssay Description:Time dependent inhibition of human recombinant MAOB at 0.25 to 1.25 uM using kynuramine substrate by fluorescence spectrophotometry based graphing of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600362(CHEMBL5187434)
Affinity DataKi:  460nMAssay Description:Time dependent inhibition of human recombinant MAOB at 0.25 to 1.25 uM using kynuramine substrate by fluorescence spectrophotometry based L-B plot an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600362(CHEMBL5187434)
Affinity DataIC50: 721nMAssay Description:Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50172756(N-benzyl-N-methylprop-2-yn-1-amine | Eutonyl | Ben...)
Affinity DataIC50: 782nMAssay Description:Inhibition of human recombinant MAOB using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50110725(CHEMBL18116 | 5-(hydroxymethyl)-3-(3-methylphenyl)...)
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50600362(CHEMBL5187434)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of human recombinant MAOB using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50172756(N-benzyl-N-methylprop-2-yn-1-amine | Eutonyl | Ben...)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed