Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50017244
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50600470(CHEMBL5174034)
Affinity DataIC50: 32nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50600471(CHEMBL5204448)
Affinity DataIC50: 69nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50314406(8-(morpholin-4-yl)-11-thia-9,14,16-triazatetracycl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50600472(CHEMBL5194579)
Affinity DataIC50: 230nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50053584(CHEMBL1977874)
Affinity DataIC50: 420nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50375667(TX-1918 | CHEMBL437612)
Affinity DataIC50: 440nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50464814(CHEMBL4281348)
Affinity DataIC50: 760nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50555900(CHEMBL4776943)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Ningbo University

Curated by ChEMBL
LigandPNGBDBM50284772(CHEMBL4161771)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed