Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50017878
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605739BDBM50605739(CHEMBL5199685)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605736BDBM50605736(CHEMBL5197084)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605734BDBM50605734(CHEMBL5185339)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605723BDBM50605723(CHEMBL5176173)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605733BDBM50605733(CHEMBL5194157)
Affinity DataIC50: 75nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605729BDBM50605729(CHEMBL5182399)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605728BDBM50605728(CHEMBL5178431)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605735BDBM50605735(CHEMBL5190284)
Affinity DataIC50: 81nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605730BDBM50605730(CHEMBL5174097)
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605737BDBM50605737(CHEMBL5177563)
Affinity DataIC50: 96nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605738BDBM50605738(CHEMBL5209397)
Affinity DataIC50: 104nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605719BDBM50605719(CHEMBL5206315)
Affinity DataIC50: 112nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605745BDBM50605745(CHEMBL5195098)
Affinity DataIC50: 134nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605732BDBM50605732(CHEMBL5194000)
Affinity DataIC50: 134nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605722BDBM50605722(CHEMBL5208801)
Affinity DataIC50: 144nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605716BDBM50605716(CHEMBL5169782)
Affinity DataIC50: 155nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605725BDBM50605725(CHEMBL5175354)
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605720BDBM50605720(CHEMBL5188393)
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605721BDBM50605721(CHEMBL5180489)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605717BDBM50605717(CHEMBL5188999)
Affinity DataIC50: 205nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605727BDBM50605727(CHEMBL5196466)
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 62810BDBM62810(2-azanyl-6-methyl-4-pyridin-3-yl-5,6,7,8-tetrahydr...)
Affinity DataIC50: 211nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605726BDBM50605726(CHEMBL5174635)
Affinity DataIC50: 214nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605715BDBM50605715(CHEMBL5196442)
Affinity DataIC50: 234nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605731BDBM50605731(CHEMBL5181302)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605724BDBM50605724(CHEMBL5198747)
Affinity DataIC50: 530nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605714BDBM50605714(CHEMBL5181742)
Affinity DataIC50: 548nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605743BDBM50605743(CHEMBL5175136)
Affinity DataIC50: 947nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605744BDBM50605744(CHEMBL5193697)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605740BDBM50605740(CHEMBL5177445)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605741BDBM50605741(CHEMBL5188825)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605718BDBM50605718(CHEMBL5194811)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605742BDBM50605742(CHEMBL5179301)
Affinity DataIC50: 3.65E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetCyclin-C(Human)
Anhui Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140257BDBM50140257(CHEMBL16171 | 5,7-Dihydroxy-8-methoxy-2-phenyl-chr...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of recombinant full length His tagged human CDK8/Cyclin C expressed in Baculovirus incubated for 60 mins in presence of ATP by ADP-Glo kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed